{"id":232147,"date":"2022-01-21T06:48:38","date_gmt":"2022-01-20T22:48:38","guid":{"rendered":"\/\/m.iemloyee.com\/?p=232147"},"modified":"2022-01-20T20:48:55","modified_gmt":"2022-01-20T12:48:55","slug":"%e5%9b%bd%e5%ae%b6%e7%ba%b3%e7%b1%b3%e7%a7%91%e5%ad%a6%e4%b8%ad%e5%bf%83%e6%9c%80%e6%96%b0angew%ef%bc%9a%e5%a4%9a%e8%82%bd%e5%8e%9f%e4%bd%8d%e8%87%aa%e7%bb%84%e8%a3%85%e7%ad%96%e7%95%a5%e7%94%a8","status":"publish","type":"post","link":"\/\/m.iemloyee.com\/?p=232147","title":{"rendered":"\u56fd\u5bb6\u7eb3\u7c73\u79d1\u5b66\u4e2d\u5fc3\u6700\u65b0Angew\uff1a\u591a\u80bd\u539f\u4f4d\u81ea\u7ec4\u88c5\u7b56\u7565\u7528\u4e8e\u764c\u75c7\u514d\u75ab\u6cbb\u7597"},"content":{"rendered":"

\u3010\u80cc\u666f\u4ecb\u7ecd\u3011<\/strong><\/p>\n

\u7efc\u5408\u4fe1\u53f7\u901a\u8def\u63a7\u5236\u7684\u751f\u7269\u5b66\u6d3b\u52a8\u7ecf\u5e38\u901a\u8fc7\u86cb\u767d\u8d28\u590d\u5408\u7269\u6784\u8c61\u7684\u5f62\u6210\uff08\u5982\u708e\u6027\u5c0f\u4f53\u7684\u7ec4\u88c5\uff09\u88ab\u6fc0\u6d3b\u7684\u3002\u7814\u7a76\u663e\u793a\uff0c\u8fd9\u4e9b\u86cb\u767d\u8d28\u590d\u5408\u7269\u7684\u4ea7\u751f\u4e25\u91cd\u4f9d\u8d56\u4e8e\u5176\u4ed6\u751f\u5316\u5206\u5b50\u7684\u8bc6\u522b\u548c\u6fc0\u6d3b\uff0c\u800c\u5728\u751f\u7406\u73af\u5883\u4e2d\u5bf9\u86cb\u767d\u8d28\u7684\u7ec4\u88c5\u72b6\u6001\u8fdb\u884c\u590d\u5236\u548c\u64cd\u63a7\u8fc4\u4eca\u4e3a\u6b62\u4f9d\u7136\u6781\u5177\u6311\u6218\u6027\u3002\u81ea\u4ece\u56fd\u5bb6\u7eb3\u7c73\u79d1\u5b66\u4e2d\u5fc3\u7684\u738b\u6d69\u8bfe\u9898\u7ec4\u57282015\u5e74\u9996\u6b21\u62a5\u9053\u4e86\u751f\u7269\u6d3b\u6027\u5206\u5b50\u7684\u4f53\u5185\u81ea\u7ec4\u88c5\u884c\u4e3a\u540e\uff0c\u5173\u4e8e\u751f\u7269\u6d3b\u6027\u7269\u8d28\u5728\u80bf\u7624\u4f4d\u70b9\u7684\u539f\u4f4d\u548c\u54cd\u5e94\u6027\u7ec4\u88c5\u7684\u7814\u7a76\u5f00\u59cb\u5f97\u5230\u5e7f\u6cdb\u7684\u5173\u6ce8\u3002\u7136\u800c\uff0c\u5c3d\u7ba1\u57fa\u4e8e\u4f53\u5185\u81ea\u7ec4\u88c5\u5efa\u7acb\u4e86\u9176\u54cd\u5e94\u7ec4\u88c5\u7684\u6982\u5ff5\uff0c\u4f46\u81ea\u7ec4\u88c5\u5206\u5b50\u9776\u5411\u63a7\u5236\u4f9d\u7136\u9c9c\u89c1\u62a5\u9053\u3002<\/p>\n

\u3010\u6210\u679c\u7b80\u4ecb\u3011<\/strong><\/p>\n

\u9488\u5bf9\u8fd9\u4e00\u6311\u6218\uff0c\u56fd\u5bb6\u7eb3\u7c73\u79d1\u5b66\u4e2d\u5fc3\u7684\u738b\u6d69<\/strong>\u7b49\u4eba\u62a5\u544a\u4e86\u4e00\u79cd\u53ef\u7f16\u7a0b\u591a\u80bd\u5206\u5b50\uff0c\u5176\u7531\u9776\u5411\u548c\u81ea\u7ec4\u88c5\u6a21\u5757\u4e24\u90e8\u5206\u7ec4\u6210\uff0c\u652f\u6301\u901a\u8fc7\u9776\u5411\u53d7\u4f53\u86cb\u767d\u800c\u5b9e\u73b0\u7684\u7279\u5b9a\u3001\u9ad8\u6548\u7684\u7ec4\u88c5\u7b56\u7565\u3002\u901a\u8fc7\u7ed1\u5b9a\u7ec6\u80de\u819c\u53d7\u4f53\uff0c\u591a\u80bd\u7684\u6784\u8c61\u80fd\u591f\u968f\u7740\u81ea\u7ec4\u88c5\u6d3b\u5316\u80fd\u7684\u964d\u4f4e\u800c\u8d8b\u4e8e\u7a33\u5b9a\uff0c\u4ece\u800c\u4fc3\u8fdb\u80bd-\u86cb\u767d\u590d\u5408\u7269\u4f4e\u805a\u5316\u3002 \u57fa\u4e8e\u6b64\uff0c\u7814\u7a76\u9996\u6b21\u8bbe\u8ba1\u5408\u6210\u4e86GNNQQNY-RGD\u591a\u80bd(G7-RGD)\uff0c\u901a\u8fc7\u8bc6\u522b\u6574\u5408\u7d20\u03b1V<\/sub>\u03b23<\/sub>\u53d7\u4f53\u6765\u9a8c\u8bc1\u4e0a\u8ff0\u81ea\u7ec4\u88c5\u6982\u5ff5\u7684\u53ef\u884c\u6027\u3002\u7531\u4e8e\u03b1V<\/sub>\u03b23<\/sub>\u7684\u5b58\u5728\uff0c\u6e38\u79bbG7-RGD\u7684\u4e34\u754c\u7ec4\u88c5\u6d53\u5ea6\u4ece525 \u03bcM\u51cf\u5c0f\u523033 \u03bcM\uff0c\u800c\u7531\u6b64\u751f\u6210G7-RGD \u7c07\u53ef\u9a71\u52a8\u6574\u5408\u7d20\u53d7\u4f53\u7684\u4f4e\u805a\u5316\u3002\u6700\u540e, \u7814\u7a76\u8fd8\u8bbe\u8ba1\u4e86\u53cc\u7279\u5f02\u6027\u7ec4\u88c5\u80bdantiCD3-G7- RGD\uff0c\u53ef\u6709\u6548\u9a71\u52a8CD3\u7684\u4f4e\u805a\u5316\u4ee5\u53ca\u4f34\u968f\u7684T\u7ec6\u80de\u6d3b\u5316\uff0c\u6700\u7ec8\u5b9e\u73b0T\u7ec6\u80de\u4ecb\u5bfc\u7684\u764c\u75c7\u514d\u75ab\u6cbb\u7597\u3002\u672c\u6587\u7b2c\u4e00\u4f5c\u8005\u4e3a<\/strong>Man-Di Wang<\/strong>\u4ee5\u53ca<\/strong>Gan-Tian Lv<\/strong>\uff0c\u7814\u7a76\u6210\u679c\u4ee5\u9898\u4e3a\u201cIn Situ Self-Assembly of Bispecific Peptide for Cancer Immunotherapy\u201d<\/strong>\u53d1\u5e03\u5728\u56fd\u9645\u8457\u540d\u671f\u520aAngew<\/em><\/strong>\u4e0a\u3002<\/p>\n

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\"\"<\/p>\n

\u56fe\u4e00\u3001<\/strong>\u53d7\u4f53\u4ecb\u5bfc\u7684<\/strong>G7-RGD<\/strong>\u7279\u5f02\u6027\u3001\u539f\u4f4d\u9ad8\u6548\u81ea\u7ec4\u88c5<\/strong><\/p>\n

\"\"<\/p>\n

\uff08a\uff09G7-RGD\u4e0d\u540c\u6d53\u5ea6\u4e0b\u7684ThT\u8367\u5149\u5f3a\u5ea6\uff1b<\/p>\n

\uff08b\uff09G7-RGD\u4e0e\u03b1V<\/sub>\u03b23<\/sub>\u5171\u5b75\u80b2\u540e\u7684ThT\u8367\u5149\u5f3a\u5ea6\uff1b<\/p>\n

\uff08c\uff09G7-RGD\u5728\u53cd\u5e94\u4e0d\u540c\u9636\u6bb5\u7684\u52bf\u80fd\u56fe\uff1b<\/p>\n

\uff08d\uff09ThT\u8367\u5149\u52a8\u529b\u5b66\u66f2\u7ebf\uff1b<\/p>\n

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\u8868\u4e00\u3001<\/strong>G7-RGD\u548c<\/strong>\u03b1V<\/sub>\u03b23<\/sub><\/strong>\u5728\u53cd\u5e94\u4e0d\u540c\u9636\u6bb5\u7684\u89e3\u79bb\u5e38\u6570\u548c\u5409\u5e03\u65af\u81ea\u7531\u80fd\u7ed3\u5408\u5e38\u6570<\/strong><\/p>\n

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\"\"<\/p>\n

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\uff08c\uff09\u5904\u7406\u6761\u4ef6\u4e0e\uff08a\uff09\u76f8\u540c\uff0c\u5171\u805a\u7126\u56fe\u50cf\u5c55\u73b0\u4e86\u591a\u80bd\u5728\u7ec6\u80de\u819c\u805a\u96c6\u7684\u8367\u5149\u5f3a\u5ea6\uff1b<\/p>\n

\uff08d\uff09\u4e0d\u540c\u65f6\u95f4\u70b9\u7684\u8367\u5149\u5f3a\u5ea6\u7edf\u8ba1\uff1b<\/p>\n

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\uff08f\uff09NBD-G7-RGD\u5904\u7406\u7684MCF-7\u7ec6\u80de\u7684\u5171\u805a\u7126\u56fe\u50cf<\/p>\n

\u56fe\u4e09\u3001\u901a\u8fc7\u9776\u5411\u8bf1\u5bfc\u62db\u52df\u7684\u7ec4\u88c5\u8fc7\u7a0b<\/strong><\/p>\n

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\uff08b\uff09Cy-G7\uff08\u7ea2\u8272\u4fe1\u53f7\uff09\u548cNBD-G7-RGD\uff08\u7eff\u8272\u4fe1\u53f7\uff09\u5728MCF-7\u7ec6\u80de\u4e0a\u7684\u5171\u5b9a\u4f4d\uff1b<\/p>\n

\uff08c\uff09\uff08b\uff09\u4e2d\u767d\u7ebf\u7684\u5f52\u4e00\u5316\u8367\u5149\u5f3a\u5ea6<\/p>\n

\u56fe\u56db\u3001<\/strong>G7-RGD<\/strong>\u81ea\u7ec4\u88c5\u8c03\u8282\u53d7\u4f53\u6574\u5408\u7d20<\/strong>\u03b1V<\/sub>\u03b23<\/sub><\/strong>\u7684\u4f4e\u805a\u5316<\/strong><\/p>\n

\u00a0\"\"<\/strong><\/p>\n

\uff08a\uff09G7-RGD\u8367\u5149\u4fe1\u53f7\u7684\u5171\u805a\u7126\u56fe\u50cf\uff1b<\/p>\n

\uff08b\uff09\u6dfb\u52a0\u591a\u80bd\u540e\u9633\u6027\u7ec6\u80de\u7684NBD\u8367\u5149\u6d41\u5f0f\u5206\u6790\uff1b<\/p>\n

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\u56fe\u4e94\u3001<\/strong>G7-antiCD3<\/strong>\u81ea\u7ec4\u88c5\u8c03\u8282\u53d7\u4f53<\/strong>CD3<\/strong>\u7684\u4f4e\u805a\u5316<\/strong><\/p>\n

\u00a0\"\"<\/strong><\/p>\n

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\uff08b\uff09\u6d41\u5f0f\u5206\u6790\u663e\u793a\u968f\u7740\u591a\u80bd\u7684\u52a0\u5165\uff0cCD3+<\/sup> T\u7ec6\u80de\u4e0a\u7684NBD\u8367\u5149\u4fe1\u53f7\u4e5f\u5f97\u5230\u4e86\u52a0\u5f3a\uff1b<\/p>\n

\uff08c\uff09CD3+<\/sup> T\u7ec6\u80de\u548cCD3–<\/sup> MCF-7 \u7ec6\u80de\u4e2dNBD+<\/sup>\u7ec6\u80de\u7684\u5360\u6bd4\uff1b<\/p>\n

\uff08d\uff09\u7531CD3-EGFP\u8f6c\u5bfc\u7684MCF-7\u7ec6\u80de\u7684\u5171\u805a\u7126\u56fe\u50cf<\/p>\n

\u56fe\u516d\u3001<\/strong>AntiCD3-G7-RGD<\/strong>\u4f5c\u4e3a\u53cc\u7279\u5f02\u6027\u5076\u8054\u7269\u6fc0\u6d3b\u5c0f\u9f20<\/strong>T<\/strong>\u7ec6\u80de<\/strong><\/p>\n

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\uff08b\uff09\u6d41\u5f0f\u5206\u6790\u6d4b\u91cf\u52a0\u5165antiCD3-G7-RGD\u540e\u7684NBD\u8367\u5149\u4fe1\u53f7\uff1b<\/p>\n

\uff08c\uff09antiCD3-G7-RGD\u5728T\u7ec6\u80de\u819c\u4e0a\u805a\u96c6\u5f62\u6210\u7eb3\u7c73\u7ea4\u7ef4\u7684SEM\u56fe\u50cf\uff1b<\/p>\n

\uff08d\uff09\u5229\u7528antiCD3-G7-RGD\u523a\u6fc0\u540e\u7684ELISA\u6d4b\u91cf\uff1b<\/p>\n

\uff08e\uff09\u6d41\u5f0f\u5206\u6790\u8868\u8fbe\u5728T\u7ec6\u80de\u8868\u9762\u7684CD69\uff1b<\/p>\n

\uff08f\uff09\u6d41\u5f0f\u5206\u6790\u8868\u8fbe\u5728T\u7ec6\u80de\u8868\u9762\u7684CD44<\/p>\n

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\"\"<\/p>\n

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\uff08b\uff09\u57fa\u4e8e\u4e73\u9178\u8131\u6c22\u9176\u6d4b\u91cfB16F10\u80bf\u7624\u7ec6\u80de\u7684\u7ec6\u80de\u6bd2\u6027<\/p>\n

\u4e0a\u8ff0\u56fe\u7247\u7248\u6743\u65b9 \u00a9 Wiley-VCH GmbH, Weinheim<\/span><\/p>\n

\u3010\u5c0f\u7ed3\u3011<\/strong><\/p>\n

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\u6587\u732e\u94fe\u63a5\uff1a<\/strong>In Situ Self-Assembly of Bispecific Peptide for Cancer Immunotherapy<\/a>, Angew<\/em>, 2021<\/strong>, DOI: 10.1002\/anie.202113649.<\/p>\n","protected":false},"excerpt":{"rendered":"

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