{"id":178354,"date":"2019-06-20T06:18:17","date_gmt":"2019-06-19T22:18:17","guid":{"rendered":"\/\/m.iemloyee.com\/?p=178354"},"modified":"2019-06-20T14:29:45","modified_gmt":"2019-06-20T06:29:45","slug":"chem-soc-rev-%e6%ad%a3%e5%b0%81%e9%9d%a2%ef%bc%9a%e6%96%b0%e5%85%b4%e7%9a%84%e5%8d%95%e5%85%83%e7%b4%a0%e4%ba%8c%e7%bb%b4%e6%9d%90%e6%96%99%e7%94%a8%e4%ba%8e%e7%94%9f%e7%89%a9%e5%8c%bb%e5%ad%a6","status":"publish","type":"post","link":"\/\/m.iemloyee.com\/?p=178354","title":{"rendered":"Chem. Soc. Rev.\u6b63\u5c01\u9762\uff1a\u65b0\u5174\u7684\u5355\u5143\u7d20\u4e8c\u7ef4\u6750\u6599\u7528\u4e8e\u751f\u7269\u533b\u5b66\u5e94\u7528"},"content":{"rendered":"

\u7814\u7a76\u80cc\u666f\u3011<\/strong><\/p>\n

\u65b0\u5174\u7684\u5355\u5143\u7d20\u4e8c\u7ef4\u6750\u6599\uff08Xenes\uff09\u5728\u5f88\u591a\u65b0\u5174\u6280\u672f\u9886\u57df\u4ee5\u53ca\u57fa\u7840\u79d1\u5b66\u9886\u57df\u7684\u62a5\u9053\u4e2d\u90fd\u663e\u793a\u51fa\u4e86\u5de8\u5927\u7684\u6f5c\u529b\uff0c\u662f\u73b0\u4eca\u6700\u4e3a\u70ed\u95e8\u7684\u7814\u7a76\u9886\u57df\u4e4b\u4e00\u3002\u7531\u4e8eXenes\uff08\u4f8b\u5982\uff0c\u787c\u70ef\u3001\u9553\u70ef\u3001\u7845\u70ef\u3001\u9517\u70ef\u3001\u9521\u70ef\u3001\u78f7\u70ef\u3001\u7837\u70ef\u3001\u9511\u70ef\u3001\u94cb\u70ef\u3001\u7852\u70ef\u548c\u78b2\u70ef\uff09\u5177\u6709\u826f\u597d\u7684\u7269\u7406\u3001\u5316\u5b66\u3001\u7535\u5b50\u548c\u5149\u5b66\u6027\u80fd\uff0c\u8fd1\u5e74\u6765\u5176\u5728\u751f\u7269\u4f20\u611f\u5668\u3001\u751f\u7269\u6210\u50cf\u3001\u836f\u7269\u9012\u9001\u548c\u75be\u75c5\u8bca\u7597\u7b49\u751f\u7269\u533b\u5b66\u9886\u57df\u5f97\u5230\u4e86\u8fc5\u731b\u5730\u53d1\u5c55\u3002\u6b64\u5916\uff0c\u7531\u4e8e\u5176\u5316\u5b66\u7ec4\u6210\u7b80\u5355\uff08\u5355\u4e00\u5143\u7d20\uff09\uff0c\u56e0\u6b64\u5bf9\u6bd4\u4e8e\u5176\u4ed6\u591a\u5143\u7d20\u7684\u4e8c\u7ef4\u6750\u6599\u53ef\u80fd\u5b58\u5728\u6613\u4e8e\u5316\u5b66\u5408\u6210\u3001\u5728\u751f\u7269\u7cfb\u7edf\u4e2d\u66f4\u5bb9\u6613\u4ee3\u8c22\u548c\u964d\u89e3\u7b49\u65b9\u9762\u7684\u6f5c\u5728\u72ec\u7279\u4f18\u52bf\u3002\u4f5c\u4e3a\u5feb\u901f\u53d1\u5c55\u7684\u4e8c\u7ef4\u6750\u6599\u9886\u57df\u4e2d\u4e00\u4e2a\u65b0\u7684\u72ec\u7279\u7684\u5206\u652f\u5b66\u79d1\uff0c\u65b0\u5174\u7684Xenes\u4ee3\u8868\u4e86\u4e0d\u540c\u751f\u7269\u533b\u5b66\u5e94\u7528\u9886\u57df\u4e2d\u7684\u65b0\u5951\u673a\u3002\u4ec5\u7ba1\u8fd9\u4e00\u9886\u57df\u53d1\u5c55\u8fc5\u901f\uff0c\u4f46\u73b0\u4eca\u53ea\u6709\u6709\u9650\u7684<\/strong>\u7efc\u8ff0\u5bf9\u65b0\u5174Xenes\u7684\u5408\u6210\u65b9\u6cd5<\/strong>\u8fdb\u884c\u4e86\u7cfb\u7edf\u603b\u7ed3\uff08Nature Reviews Chemistry<\/em><\/strong> 2017, 1, 0014; Chemical Society Reviews<\/em><\/strong> 2017, 46, 2127-2157; Nature Materials<\/em><\/strong> 2017, 16, 163-169\uff09\u3002\u76ee\u524d\uff0c\u5c1a\u6ca1\u6709\u7efc\u8ff0\u6587\u7ae0\u7cfb\u7edf\u5730\u603b\u7ed3\u3001\u5f52\u7eb3\u5404\u7c7b\u522b\u65b0\u5174Xenes\u7684\u7ed3\u6784\u548c\u529f\u80fd\u4e0e\u5176\u5bf9\u5e94\u7684\u751f\u7269\u533b\u5b66\u5e94\u7528\u4e4b\u95f4\u7684\u5173\u8054<\/strong>\u3002\uff08\u5907\u6ce8\uff1a\u77f3\u58a8\u70ef\u4e0d\u5c5e\u4e8e\u672c\u6587\u6240\u5b9a\u4e49\u7684\u65b0\u5174Xenes\u8ba8\u8bba\u8303\u56f4\u3002\uff09<\/p>\n

\u3010\u6210\u679c\u7b80\u4ecb\u3011<\/strong><\/p>\n

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\"\"<\/a><\/p>\n

TOC<\/strong>\u4ee5\u53ca\u8bba\u6587\u5c01\u9762<\/strong><\/p>\n

\u3010\u56fe\u6587\u5bfc\u8bfb\u3011<\/strong><\/p>\n

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\"\"<\/a><\/p>\n

\u56fe\u4e8c: \u65b0\u5174\u7684\u5355\u5143\u7d20\u4e8c\u7ef4\u6750\u6599\uff08Xenes\uff09\u7684\u5206\u7c7b\u7684\u5408\u6210\u65b9\u6cd5\u793a\u610f\u56fe: (a)\u81ea\u4e0b\u800c\u4e0a\u7684\u5408\u6210\u65b9\u6cd5\uff08\u4f8b\u5982\u5316\u5b66\u6c14\u76f8\u6c89\u79ef\u3001\u7269\u7406\u6c14\u76f8\u6c89\u79ef\u548c\u6e7f\u5316\u5b66\u6cd5\u7b49\uff09\uff1b (b)\u81ea\u4e0a\u800c\u4e0b\u7684\u5408\u6210\u65b9\u6cd5\uff08\u4f8b\u5982\u6db2\u76f8\u5265\u79bb\u3001\u673a\u68b0\u5265\u79bb\u548c\u8680\u523b\u7b49\uff09\u3002<\/p>\n

\"\"<\/a><\/p>\n

\u56fe\u4e09: \u5468\u671f\u8868\u5143\u7d20\u5bf9\u5e94\u7684Xenes\uff08\u7b2cIII\u65cf\u787c\u70ef\u548c\u9553\u70ef\uff1b\u7b2cIV\u65cf\u7845\u70ef\u3001\u9517\u70ef\u548c\u9521\u70ef\uff1b\u7b2cV\u65cf\u78f7\u70ef\u3001\u7837\u70ef\u3001\u9511\u70ef\u548c\u94cb\u70ef\uff1b\u7b2cVI\u65cf\u7852\u70ef\u548c\u78b2\u70ef\uff09\u53ca\u5176\u5bf9\u5e94\u7684\u5df2\u88ab\u62a5\u9053\u7684\u5408\u6210\u65b9\u6cd5\u3002\u767d\u8272\u663e\u793a\u7684\u5143\u7d20\u5bf9\u5e94\u7684Xenes\u5df2\u7ecf\u88ab\u5408\u6210\uff0c\u7070\u8272\u663e\u793a\u7684\u5143\u7d20\u5bf9\u5e94\u7684Xenes\u76ee\u524d\u8fd8\u6ca1\u6709\u88ab\u9884\u6d4b\u6216\u8005\u5b9e\u9a8c\u5ba4\u5408\u6210\u5236\u5907\u3002<\/p>\n

\"\"<\/a><\/p>\n

\u56fe\u56db: \u751f\u7269\u533b\u5b66\u5e94\u7528\u4e2d\u65b0\u5174Xenes\u8868\u9762\u529f\u80fd\u5316\u7b56\u7565\u7684\u4f8b\u5b50\u3002(a) \u78b1\u91d1\u5c5e\u5bf9\u7845\u70ef\u7684\u8868\u9762\u5438\u9644; (b)\u9511\u70ef\u7684\u805a\u4e59\u4e8c\u9187\u5316; (c)\u805a\u4e59\u70ef\u5421\u54af\u70f7\u916e\u6d82\u8986\u94cb\u70ef; (d)\u5c06\u78f7\u70ef\u5305\u5c01\u5728PLGA\u805a\u5408\u7269\u4e2d; (e)\u8c37\u80f1\u7518\u80bd\u5bf9\u78b2\u70ef\u7684\u6539\u6027\u3002<\/p>\n

\"\"<\/a><\/p>\n

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\"\"<\/a><\/p>\n

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\"\"<\/a><\/p>\n

\u56fe\u4e03: \u57fa\u4e8e\u65b0\u5174Xenes\u7684\u836f\u7269\u8f7d\u4f53\uff08\u9012\u9001\u5c0f\u5206\u5b50\u836f\u7269\u3001siRNA\u7b49\uff09\u8bbe\u8ba1\u548c\u5149\u5b66\u6cbb\u7597\uff08\u5149\u70ed\u6cbb\u7597\u3001\u5149\u52a8\u529b\u6cbb\u7597\u7b49\uff09\u5e94\u7528\u3002<\/p>\n

\"\"<\/p>\n

 <\/p>\n

\u56fe\u516b: \u57fa\u4e8e\u65b0\u5174Xenes\u7684\u8bca\u65ad\u6cbb\u7597\u5e94\u7528\u3002\u4f8b\u5982\uff0c\u57fa\u4e8e\u8d85\u5c0f\u94cb\u7eb3\u7c73\u70b9\uff08\u94cb\u70ef\uff09\u7684CT\/\u5149\u58f0\u53cc\u6210\u50cf\u5f15\u5bfc\u7684\u80bf\u7624\u5149\u70ed\u548c\u653e\u7597\u8054\u5408\u6cbb\u7597\uff1b\u57fa\u4e8e\u9511\u70ef\u7684\u5149\u58f0\/\u8367\u5149\/\u5149\u70ed\u6210\u50cf\u5f15\u5bfc\u7684\u80bf\u7624\u5149\u5408\u548c\u5316\u7597\u8054\u5408\u6cbb\u7597\u3002<\/p>\n

\"\"<\/a><\/p>\n

\u56fe\u4e5d: \u57fa\u4e8e\u65b0\u5174Xenes\u7684\u6297\u83cc\u5e94\u7528\u3001\u9aa8\u518d\u751f\u53ca\u7ec4\u7ec7\u5de5\u7a0b\u4ee5\u53ca\u795e\u7ecf\u9000\u884c\u6027\u75be\u75c5\u6cbb\u7597\u7b49\u3002<\/p>\n

\"\"<\/a><\/p>\n

\u3010\u603b\u7ed3\u5c55\u671b\u3011<\/strong><\/p>\n

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\u867d\u7136\u8bb8\u591a\u7814\u7a76\u8868\u660eXenes\u5728\u751f\u7269\u533b\u5b66\u5e94\u7528\u4e2d\u5177\u6709\u5de8\u5927\u6f5c\u529b\uff0c\u4f46\u5176\u76f8\u5bf9\u4e0d\u53ef\u63a7\u7684\u5f62\u6001\u548c\u8f83\u5bbd\u7684\u5c3a\u5bf8\u5206\u5e03\u53ef\u80fd\u4f1a\u5bf9\u5176\u66f4\u8fdb\u4e00\u6b65\u5730\u53d1\u5c55\u5b58\u5728\u9650\u5236\u3002\u6b64\u5916\uff0c\u5728\u83b7\u5f97\u76d1\u7ba1\u673a\u6784\u6279\u51c6\u4e4b\u524d\uff0c\u5e94\u59cb\u7ec8\u8003\u8651\u5e76\u89e3\u51b3Xenes\u7eb3\u7c73\u5e73\u53f0\u5728\u533b\u836f\u9886\u57df\u4e2d\u7684\u6f5c\u5728\u6bd2\u6027\u3002\u56e0\u6b64\uff0c\u4e00\u4e9b\u4f5c\u8005\u63cf\u8ff0\u4e86\u5b9a\u4e49\u5b89\u5168\u7b49\u7ea7\u7684\u5341\u591a\u4e2a\u5173\u952e\u56e0\u7d20\uff0c\u4ee5\u8bc4\u4f30\u65b0\u7eb3\u7c73\u6750\u6599\u7684\u6f5c\u5728\u6bd2\u6027\u3002\u7136\u800c\uff0cXenes\u7684\u8868\u5f81\u53ef\u80fd\u5728\u751f\u7269\u6d4b\u8bd5\u671f\u95f4\u6539\u53d8\uff0c\u8fd9\u4f7f\u5f97\u5728\u76f8\u540c\u5b9e\u9a8c\u6761\u4ef6\u4e0b\u8fdb\u884c\u7684Xenes\u7684\u7269\u7406\u5316\u5b66\u8868\u5f81\u66f4\u590d\u6742\u3002\u5728\u6b64\u57fa\u7840\u4e0a\uff0c\u5e94\u63d0\u51fa\u4e00\u4e2a\u89c4\u5219\uff0c\u5176\u4e2d\u5305\u542b\u4e00\u4e9b\u5173\u952e\u56e0\u7d20\uff0c\u4ee5\u6807\u51c6\u5316\u6bd4\u8f83\u7279\u5f81\u548c\u7ed3\u679c\u7684\u65b9\u6cd5\u3002\u7814\u7a76\u4eba\u5458\u5df2\u671d\u7740\u8fd9\u4e2a\u65b9\u5411\u505a\u51fa\u4e86\u4e00\u4e9b\u52aa\u529b\uff0c\u5e76\u63d0\u51fa\u4e86\u4e00\u4e9b\u7eb3\u7c73\u6750\u6599\u7279\u6027\u7684\u534f\u8bae\uff0c\u5305\u62ec\u6750\u6599\u7684\u5408\u6210\u8fc7\u7a0b\u548c\u751f\u7269\u6d4b\u8bd5\u3002\u6b64\u5916\uff0c\u867d\u7136Xenes\u5728\u751f\u7269\u7cfb\u7edf\u4e2d\u66f4\u5bb9\u6613\u7684\u4ee3\u8c22\u548c\u964d\u89e3\u7684\u4f18\u52bf\uff0cXenes\u7684\u7eb3\u7c73\u6750\u6599-\u751f\u7269\u76f8\u4e92\u4f5c\u7528\u4ecd\u7136\u9700\u8981\u88ab\u6df1\u5165\u7814\u7a76\u3002\u5c3d\u7ba1\u4e00\u4e9bXenes\u7684\u751f\u7269\u533b\u5b66\u5e94\u7528\u5df2\u88ab\u5e7f\u6cdb\u7814\u7a76\uff08\u5982\u78f7\u70ef\uff09\uff0c\u4f46\u4e00\u4e9b\u65b0\u5408\u6210\u7684Xenes\u4ecd\u7136\u5904\u4e8e\u5176\u751f\u7269\u5e94\u7528\u7684\u5f00\u59cb\u9636\u6bb5\uff08\u4f8b\u5982\uff0c\u9553\u70ef\u3001\u9517\u70ef\u3001\u9521\u70ef\u3001\u7837\u70ef\u548c\u7852\u70ef\uff09\uff0c\u8fd9\u610f\u5473\u7740\u5728\u4e0d\u4e45\u7684\u5c06\u6765\uff0c\u8fd9\u4e9bXenes\u5c06\u53ef\u80fd\u627e\u5230\u66f4\u591a\u7684\u5e94\u7528\u673a\u4f1a\u3002<\/p>\n

\u5728Xenes\u7684\u8868\u5f81\u4e2d\u5fc5\u987b\u8003\u8651\u4e00\u4e9b\u7269\u7406\u5316\u5b66\u6027\u8d28\uff0c\u5305\u62ec\u5c42\u6570\uff0c\u6c27\u5316\u7a0b\u5ea6\u548c\u6a2a\u5411\u5c3a\u5bf8\u3002\u6b64\u5916\uff0c\u6613\u805a\u96c6\uff0c\u5feb\u901f\u964d\u89e3\u548c\u7a33\u5b9a\u6027\u4e0d\u8db3\u7b49\u7f3a\u70b9\u4e5f\u9650\u5236\u4e86Xenes\u5728\u751f\u7269\u73af\u5883\u4e2d\u7684\u5e94\u7528\uff0c\u8fd9\u4e2a\u95ee\u9898\u5e94\u8be5\u8fdb\u4e00\u6b65\u89e3\u51b3\u3002\u8fd8\u5e94\u6ce8\u610f\uff0cXenes\u964d\u89e3\u7684\u56e0\u7d20\u6709\u4e24\u4e2a\u65b9\u9762\uff1a\u8fc7\u5feb\u7684\u964d\u89e3\u5c06\u9650\u5236\u5f00\u53d1\u7684Xenes\u7684\u6cbb\u7597\u6548\u679c\uff0c\u800c\u5b83\u4eec\u7684\u964d\u89e3\u6027\u5728\u751f\u7269\u533b\u5b66\u5e94\u7528\u4e2d\u662f\u9700\u8981\u7684\u3002\u56e0\u6b64\uff0c\u5236\u5907\u5177\u6709\u53ef\u8c03\u8282\u964d\u89e3\u901f\u7387\u7684\u529f\u80fd\u5316Xenes\u5bf9\u4e8e\u6700\u4f73\u6cbb\u7597\u529f\u6548\u548c\u6700\u4f4e\u5168\u8eab\u6bd2\u6027\u4e5f\u662f\u91cd\u8981\u7684\u3002\u5bf9\u4e8eXenes\u800c\u8a00\uff0c\u5b83\u4eec\u5728\u5206\u6563\u4f53\u4e2d\u7684\u521d\u59cb\u7ed3\u6784\u7279\u5f81\u5728\u51e0\u5c0f\u65f6\u751a\u81f3\u4e00\u5929\u6216\u66f4\u957f\u65f6\u95f4\u540e\u53ef\u80fd\u662f\u4e0d\u4e00\u6837\u7684\uff0c\u56e0\u6b64\u627e\u51fa\u60ac\u6d6e\u6db2\u7684\u53d8\u5316\u5e76\u5c06\u5176\u5e94\u7528\u4e8e\u751f\u7406\u5b9e\u9a8c\u662f\u975e\u5e38\u91cd\u8981\u7684\u3002\u56e0\u6b64\uff0cXenes\u6c34\u6eb6\u6db2\u7684\u5206\u6563\u6027\u548c\u7a33\u5b9a\u6027\u662f\u751f\u7269\u5b9e\u9a8c\u7684\u9996\u8981\u4efb\u52a1\u3002\u63d0\u9ad8\u5176\u5206\u6563\u6027\u548c\u7a33\u5b9a\u6027\u5bf9\u4e8e\u63a8\u8fdb\u4e0d\u540c\u7684\u751f\u7269\u533b\u5b66\u5e94\u7528\u81f3\u5173\u91cd\u8981\u3002\u9664\u6b64\u4e4b\u5916\uff0c\u7814\u7a76\u4eba\u5458\u5f00\u53d1\u4e86\u5f88\u591a\u65b9\u6cd5\u6765\u5bf9Xenes\u8fdb\u884c\u6539\u6027\uff0c\u4ee5\u5728\u751f\u7269\u533b\u5b66\u5e94\u7528\u7684\u60ac\u6d6e\u6db2\u4e2d\u83b7\u5f97\u7a33\u5b9a\u7684\u7247\u6750\u3002\u65e0\u8bbaXenes\u56fa\u6709\u7684\u751f\u7269\u76f8\u5bb9\u6027\u5982\u4f55\uff0c\u90fd\u5e94\u7cbe\u786e\u91cf\u5316\u5b83\u4eec\u7684\u5206\u6563\uff0c\u4ee5\u5c3d\u91cf\u51cf\u5c11\u53ef\u80fd\u7684\u751f\u7269\u6548\u5e94\uff0c\u4ece\u800c\u8fdb\u4e00\u6b65\u4e86\u89e3\u5b83\u4eec\u7684\u771f\u6b63\u4f5c\u7528\u3002<\/p>\n

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\u3010\u901a\u8baf\u4f5c\u8005\u4ecb\u7ecd\u3011<\/strong><\/p>\n

\u9676\u4f1f<\/strong>\u535a\u58eb\u4e8e2015\u5e747\u6708\u5728\u6e05\u534e\u5927\u5b66\u83b7\u5f97\u7406\u5b66\u535a\u58eb\u5b66\u4f4d\u3002\u968f\u540e\uff0c\u4ed6\u5728\u54c8\u4f5b\u5927\u5b66\u533b\u5b66\u9662Omid C. Farokhzad\u6559\u6388\u56e2\u961f\u62c5\u4efbNIH\u8d44\u52a9\u7684\u535a\u58eb\u540e\u7814\u7a76\u5458\uff0c\u5e76\u4e8e2018\u5e743\u6708\u53d7\u8058\u4e3a\u54c8\u4f5b\u5927\u5b66\u533b\u5b66\u9662\u8bb2\u5e08\u3002\u7814\u7a76\u65b9\u5411\u4e3b\u8981\u5305\u62ec\u529f\u80fd\u7eb3\u7c73\u6750\u6599\u7684\u8bbe\u8ba1\u548c\u5408\u6210\uff0c\u63a2\u7d22\u5b83\u4eec\u7684\u4f53\u5185\u4ea4\u4e92\u4f5c\u7528\u673a\u5236\u548c\u5e7f\u6cdb\u7684\u751f\u7269\u533b\u5b66\u5e94\u7528\uff08\u5982RNA\u9012\u9001\u3001\u764c\u75c7\u8bca\u65ad\u6cbb\u7597\u3001\u4f24\u53e3\u6108\u5408\u3001\u5fc3\u8840\u7ba1\u75be\u75c5\u548c\u7cd6\u5c3f\u75c5\u6cbb\u7597\uff09\u3002\u5728Nature Biomedical Engineering<\/em>, Nature Communications<\/em>, Chemical Society Reviews<\/em>, Advanced Materials<\/em>, Angewandte Chemie<\/em>, ACS Nano<\/em>, Nano Letters<\/em>\u7b49\u520a\u7269\u4e0a\u53d1\u8868\u8bba\u658760\u4f59\u7bc7\uff08\u5176\u4e2d\u5c01\u9762\u8bba\u658715\u7bc7\uff0cESI\u9ad8\u5f15\u7528\u524d1%\u8bba\u658710\u7bc7\uff0c\u70ed\u95e8\u8bba\u6587\u524d0.1%\u8bba\u65872\u7bc7\uff09\u3002\u4ed6\u662fFrontiers\u7f16\u8f91\u59d4\u5458\u4f1a\u6210\u5458\uff0cFrontiers in Pharmacology<\/em>\u6742\u5fd7\u5ba2\u5ea7\u4e3b\u7f16\u3002\u9676\u4f1f\u535a\u58eb\u66fe\u83b7\u5f97\u7f8e\u56fdMETAvivor\u9752\u5e74\u7814\u7a76\u5458\u5956\u3001\u54c8\u4f5b\u5927\u5b66\u533b\u5b66\u9662\u9ebb\u9189\u7cfb\u57fa\u7840\u79d1\u5b66\u5bb6\u57fa\u91d1\u3001\u7f8e\u56fd\u5fc3\u810f\u534f\u4f1a\u5408\u4f5c\u79d1\u5b66\u5956\u7b49\u5956\u9879\/\u57fa\u91d1\u3002<\/p>\n

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