{"id":151711,"date":"2018-08-26T06:13:41","date_gmt":"2018-08-25T22:13:41","guid":{"rendered":"\/\/m.iemloyee.com\/?p=151711"},"modified":"2018-08-25T17:14:16","modified_gmt":"2018-08-25T09:14:16","slug":"%e4%b8%ad%e7%a7%91%e9%99%a2%e8%bf%87%e7%a8%8b%e6%89%80%e9%97%ab%e5%ad%a6%e6%b5%b7-jacs-%e5%a4%9a%e7%bb%84%e5%88%86%e9%85%8d%e4%bd%8d%e8%87%aa%e7%bb%84%e8%a3%85%e8%ae%be%e8%ae%a1%e7%9a%84%e6%99%ba","status":"publish","type":"post","link":"\/\/m.iemloyee.com\/?p=151711","title":{"rendered":"\u4e2d\u79d1\u9662\u8fc7\u7a0b\u6240\u95eb\u5b66\u6d77 JACS: \u591a\u7ec4\u5206\u914d\u4f4d\u81ea\u7ec4\u88c5\u8bbe\u8ba1\u7684\u667a\u80fd\u80bd\u57fa\u8d85\u5206\u5b50\u5149\u52a8\u529b\u91d1\u5c5e\u7eb3\u7c73\u836f\u7269"},"content":{"rendered":"
\u3010\u5f15\u8a00\u3011<\/strong><\/div>\n
\u00a0<\/div>\n
\u5149\u52a8\u529b\u7597\u6cd5\uff08PDT\uff09\u662f\u4e00\u79cd\u65b0\u5174\u7684\u6cbb\u7597\u65b9\u5f0f\uff0c\u5176\u5c06\u5149\u654f\u6027\u836f\u7269\uff08\u5149\u654f\u5242\uff09\u548c\u5149\u4e0e\u5185\u6e90\u6027\u7684\u6c27\u7ed3\u5408\uff0c\u901a\u8fc7\u590d\u6742\u7684\u5149\u5316\u5b66\u548c\u751f\u7269\u7ea7\u8054\u53cd\u5e94\uff0c\u5bf9\u80bf\u7624\u53d1\u6325\u6740\u4f24\u4f5c\u7528\u3002\u7531\u4e8e\u7eb3\u7c73\u5242\u578b\u80fd\u591f\u589e\u5f3a\u836f\u7269\u7684\u80bf\u7624\u9009\u62e9\u6027\uff0c\u63d0\u9ad8\u6cbb\u7597\u7cbe\u786e\u5ea6\u548c\u6548\u7387\uff0c\u5149\u654f\u5242\u7eb3\u7c73\u836f\u7269\u7684\u7814\u7a76\u6210\u4e3a\u8fd1\u6765\u7684\u7814\u7a76\u70ed\u70b9\u3002\u7eb3\u7c73\u5149\u654f\u5242\u4f1a\u6291\u5236\u6d3b\u6027\u6c27\uff08ROS\uff09\u7684\u4ea7\u751f\uff0c\u56e0\u6b64\u9700\u8981\u5176\u5728\u76ee\u6807\u7ec6\u80de\u4e2d\u5feb\u901f\u91ca\u653e\u5149\u654f\u5242\u3002\u73b0\u6709\u7684\u5149\u654f\u5242\u7eb3\u7c73\u836f\u7269\u5177\u6709\u4ee5\u4e0b\u51e0\u4e2a\u7f3a\u70b9\uff1a\u9996\u5148\uff0c\u5c1a\u672a\u5728\u5149\u654f\u5242\u7eb3\u7c73\u836f\u7269\u4e2d\u540c\u65f6\u5b9e\u73b0\u957f\u8840\u6db2\u5faa\u73af\u65f6\u95f4\u548c\u9776\u5411\u6027\u7206\u53d1\u91ca\u653e\uff1b\u5176\u6b21\uff0c\u5e38\u89c4\u9012\u9001\u8f7d\u4f53\u5bf9\u5149\u654f\u5242\u7684\u88c5\u8f7d\u7387\u8f83\u4f4e\u4e14\u6613\u4e8e\u5728\u8840\u6db2\u4e2d\u8fc7\u65e9\u91ca\u653e\uff1b\u7b2c\u4e09\uff0c\u57fa\u4e8e\u5f31\u76f8\u4e92\u4f5c\u7528\u7684\u81ea\u7ec4\u88c5\u7eb3\u7c73\u836f\u7269\u5728\u7a00\u91ca\u65f6\u6613\u4e8e\u5feb\u901f\u89e3\u7ec4\u88c5\uff0c\u4ece\u800c\u5931\u53bb\u80bf\u7624\u7279\u5f02\u6027\u5bcc\u96c6\u80fd\u529b\uff1b\u6700\u540e\uff0c\u4e00\u4e9b\u4eba\u5de5\u5408\u6210\u5206\u5b50\u53ef\u80fd\u5f15\u8d77\u6bd2\u6027\u3001\u514d\u75ab\u548c\u708e\u75c7\u53cd\u5e94\u7b49\u526f\u4f5c\u7528\u3002\u4ee5\u751f\u7269\u5206\u5b50\u4f5c\u4e3a\u81ea\u7ec4\u88c5\u57fa\u5143\uff0c\u901a\u8fc7\u914d\u4f4d\u4f5c\u7528\u548c\u591a\u79cd\u5f31\u76f8\u4e92\u4f5c\u7528\u7684\u534f\u540c\uff0c\u6784\u7b51\u65b0\u578b\u7684\u5149\u654f\u5316\u7eb3\u7c73\u836f\u7269\uff0c\u6709\u671b\u7528\u4e8e\u89e3\u51b3\u4e0a\u8ff0\u95ee\u9898\u3002<\/div>\n
\u00a0<\/div>\n
\u3010\u6210\u679c\u7b80\u4ecb\u3011<\/strong><\/div>\n
\u00a0<\/div>\n
\u8fd1\u65e5\uff0c\u4e2d\u56fd\u79d1\u5b66\u9662\u8fc7\u7a0b\u5de5\u7a0b\u7814\u7a76\u6240\u7684\u95eb\u5b66\u6d77\u7814\u7a76\u5458\uff08\u901a\u8baf\u4f5c\u8005\uff09<\/strong>\u7b49\u62a5\u9053\u4e86\u4e00\u79cd\u591a\u7ec4\u5206\u914d\u4f4d\u81ea\u7ec4\u88c5\u7684\u7b56\u7565\uff0c\u5e76\u901a\u8fc7\u8be5\u7b56\u7565\u5b9e\u73b0\u4e86\u667a\u80fd\u8d85\u5206\u5b50\u5149\u52a8\u529b\u7eb3\u7c73\u836f\u7269\u7684\u6784\u7b51\u3002\u53d7\u91d1\u5c5e\u86cb\u767d\u4e2d\u591a\u7ec4\u5206\u76f8\u4e92\u4f5c\u7528\u7684\u542f\u53d1\uff0c\u8bbe\u8ba1\u4e86\u5177\u6709\u91d1\u5c5e\u914d\u4f4d\u80fd\u529b\u7684\u591a\u80bd\uff0c\u5e76\u901a\u8fc7\u591a\u80bd\u3001\u5149\u654f\u5242\u548c\u91d1\u5c5e\u79bb\u5b50\u7684\u534f\u540c\u4f5c\u7528\uff0c\u5236\u5907\u4e86\u5c3a\u5bf8\u5747\u4e00\u3001\u7ed3\u6784\u89c4\u6574\u3001\u5149\u654f\u5242\u88c5\u8f7d\u6548\u7387\u9ad8\u7684\u7eb3\u7c73\u836f\u7269\u3002\u5149\u654f\u5242\u7eb3\u7c73\u836f\u7269\u7684\u5f62\u6210\u8fc7\u7a0b\u4e2d\u5305\u542b\u4e86\u914d\u4f4d\u3001\u758f\u6c34\u3001\u9759\u7535\u7b49\u76f8\u4e92\u4f5c\u7528\u7684\u534f\u540c\u3002\u7a33\u5b9a\u6027\u6d4b\u8bd5\u8868\u660e\uff0c\u5149\u654f\u5242\u7eb3\u7c73\u836f\u7269\u5728\u6c34\u4f53\u7cfb\u4e2d\u80f6\u4f53\u7a33\u5b9a\u6027\u5f3a\uff0c\u5728pH\u548c\u6c27\u5316\u8fd8\u539f\u4f5c\u7528\u7684\u523a\u6fc0\u4e0b\u80fd\u591f\u7206\u53d1\u6027\u91ca\u653e\u5149\u654f\u5242\u3002\u4f53\u5185\u5b9e\u9a8c\u8bc1\u5b9e\u7eb3\u7c73\u836f\u7269\u6709\u6548\u5730\u5ef6\u957f\u4e86\u5149\u654f\u5242\u7684\u8840\u6db2\u5faa\u73af\u65f6\u95f4\u3001\u589e\u5f3a\u4e86\u5149\u654f\u5242\u7684\u80bf\u7624\u5bcc\u96c6\u6548\u679c\uff0c\u6700\u7ec8\u5b9e\u73b0\u4e86\u9ad8\u6548\u7684\u5149\u52a8\u529b\u6297\u80bf\u7624\u6cbb\u7597\u3002\u672c\u7814\u7a76\u63d0\u4f9b\u4e86\u4e00\u79cd\u65b0\u578b\u7684\u7eb3\u7c73\u836f\u7269\u5236\u5907\u7b56\u7565\uff0c\u8fd9\u79cd\u7b56\u7565\u666e\u904d\u9002\u7528\u4e8e\u589e\u5f3a\u5149\u654f\u5242\u7684\u80bf\u7624\u7279\u5f02\u6027\u9012\u9001\u548c\u6cbb\u7597\uff0c\u4e3a\u5f00\u53d1\u4e0b\u4e00\u4ee3\u667a\u80fd\u5149\u654f\u7eb3\u7c73\u836f\u7269\u63d0\u4f9b\u4e86\u65b0\u7684\u542f\u793a\u3002\u7814\u7a76\u6210\u679c\u4ee5\u9898\u4e3a\u201cSmart Peptide-Based Supramolecular Photodynamic Metallo Nanodrugs Designed by Multicomponent Coordination Self-Assembly\u201d<\/strong>\u53d1\u5e03\u5728\u56fd\u9645\u8457\u540d\u671f\u520aJACS<\/strong>\u4e0a\u3002<\/div>\n
\u00a0<\/div>\n
\u3010\u56fe\u6587\u5bfc\u8bfb\u3011<\/strong><\/div>\n
\u00a0<\/div>\n
\u56fe\u4e00\u3001\u7528\u4e8e\u6709\u6548\u6297\u80bf\u7624PDT\u7684\u8d85\u5206\u5b50\u91d1\u5c5e\u7eb3\u7c73\u836f\u7269\u7684\u793a\u610f\u56fe\"\"<\/strong><\/div>\n
\u00a0<\/div>\n
\uff08a\uff09 \u4eba\u8840\u7ea2\u86cb\u767d\u4e2d\u8840\u7ea2\u7d20\u57fa\u56e2\u548c\u7ec4\u6c28\u9178\u4e0e\u91d1\u5c5e\u79bb\u5b50\u7684\u534f\u540c\u914d\u4f4d\u4f5c\u7528\uff1b<\/div>\n
\u00a0<\/div>\n
\uff08b\uff09 \u950c\u79bb\u5b50\u534f\u540c\u914d\u4f4d\u77ed\u80bd\u548c\u5149\u654f\u5242\u6784\u5efa\u91d1\u5c5e\u7eb3\u7c73\u836f\u7269\uff1b<\/div>\n
\u00a0<\/div>\n
\uff08c\uff09 \u7ec4\u88c5\u4f53\u4e2d\u950c\u79bb\u5b50\u4e0e\u77ed\u80bd\u7684\u5206\u5b50\u7ec4\u7ec7\u6a21\u5f0f\uff1b<\/div>\n
\u00a0<\/div>\n
\uff08d\uff09 \u91d1\u5c5e\u7eb3\u7c73\u836f\u7269\u901a\u8fc7\u8840\u6db2\u5faa\u73af\u5728\u80bf\u7624\u4e2d\u5bcc\u96c6\uff1b<\/div>\n
\u00a0<\/div>\n
\uff08e\uff09 \u91d1\u5c5e\u7eb3\u7c73\u836f\u7269\u901a\u8fc7\u80de\u541e\u4f5c\u7528\u8fdb\u5165\u80bf\u7624\u7ec6\u80de\uff0c\u5728\u7ec6\u80de\u5fae\u73af\u5883\u7684\u4f5c\u7528\u4e0b\u7a81\u91ca\u5149\u654f\u5242\uff0c\u91ca\u653e\u7684\u5149\u654f\u5242\u5728\u5149\u7684\u4f5c\u7528\u4e0b\u4ea7\u751fPDT\u4f5c\u7528\u3002<\/div>\n
\u00a0<\/div>\n
\u56fe\u4e8c\u3001Fmoc-H \/ Zn2+<\/sup>\u548cZ-HF \/ Zn2+<\/sup>\u7eb3\u7c73\u9897\u7c92\u7684\u5f62\u6001\u3001\u914d\u4f4d\u6a21\u5f0f\u3001FTIR\u5149\u8c31\u548c\u8d85\u7075\u654f\u54cd\u5e94\u6027\"\"<\/strong><\/div>\n
\u00a0<\/div>\n
\uff08a\uff09 Fmoc-H \/ Zn2+<\/sup>\u548cZ-HF \/ Zn2+<\/sup> \u7684DLS\u548c\u6837\u54c1\u7684\u56fe\u7247\uff1b<\/div>\n
\u00a0<\/div>\n
\uff08b\uff09 Fmoc-H \/ Zn2+<\/sup>\u548cZ-HF \/ Zn2+<\/sup>\u7684SEM\u56fe\uff1b<\/div>\n
\u00a0<\/div>\n
\uff08c\uff09 Fmoc-H \/ Zn2+<\/sup>\u548cZ-HF \/ Zn2+<\/sup>\u7684TEM\u56fe\uff1b<\/div>\n
\u00a0<\/div>\n
\uff08d\uff09 Fmoc-H \/ Zn2+<\/sup>\u7eb3\u7c73\u9897\u7c92\u4e2d\u80bd\u548cZn2+<\/sup>\u7684\u7a7a\u95f4\u914d\u4f4d\u6784\u8c61\u4ee5\u53ca\u914d\u4f4d\u952e\u7684\u957f\u5ea6\uff1b<\/div>\n
\u00a0<\/div>\n
\uff08e\uff09 \u5b9e\u9a8c\u548c\u8ba1\u7b97\u7684Fmoc-H \/ Zn2+<\/sup>\u548cZ-HF \/ Zn2+<\/sup>\u7684FTIR\u5149\u8c31\uff1b<\/div>\n
\u00a0<\/div>\n
\uff08f, g\uff09Fmoc-H \/ Zn2+<\/sup>\u5bf9pH\u548cGSH\u53d8\u5316\u7684\u8d85\u7075\u654f\u54cd\u5e94\u7684\u793a\u610f\u56fe\u548c\u56fe\u7247\u3002<\/div>\n
\u00a0<\/div>\n
\u56fe\u4e09\u3001\u91d1\u5c5e\u7eb3\u7c73\u836f\u7269\u7684\u5f62\u8c8c\u3001\u7d2b\u5916-\u53ef\u89c1\u5438\u6536\u5149\u8c31\u3001\u7a33\u5b9a\u6027\u548c\u54cd\u5e94\"\"<\/strong><\/div>\n
\u00a0<\/div>\n
\uff08a\uff09 Fmoc-H \/ Zn2+<\/sup> \/ Ce6\u548cZ-HF \/ Zn2+<\/sup> \/ Ce6\u7684DLS\u548c\u6837\u54c1\u7684\u56fe\u7247\uff1b<\/div>\n
\u00a0<\/div>\n
\uff08b\uff09 Fmoc-H \/ Zn2+<\/sup> \/ Ce6\u548cZ-HF \/ Zn2+<\/sup> \/ Ce6\u7684SEM\u56fe\uff1b<\/div>\n
\u00a0<\/div>\n
\uff08c\uff09 Fmoc-H \/ Zn2+<\/sup> \/ Ce6\u548cZ-HF \/ Zn2+<\/sup> \/ Ce6\u7684TEM\u56fe\uff1b<\/div>\n
\u00a0<\/div>\n
\uff08d\uff09 Fmoc-H \/ Zn2+<\/sup> \/ Ce6\u3001Z-HF \/ Zn2+<\/sup> \/ Ce6\u3001\u5355\u4f53Ce6\u548cCe6\u805a\u96c6\u4f53\u7684\u7d2b\u5916-\u53ef\u89c1\u5438\u6536\u56fe\uff1b<\/div>\n
\u00a0<\/div>\n
\uff08e\uff09 \u7a00\u91ca\u7684Fmoc-H \/ Zn2+<\/sup> \/ Ce6\u548cZ-HF \/ Zn2+<\/sup> \/ Ce6\u572837 \u2103\u4e0b\u5b75\u80b2\u65f6\u7684\u5c3a\u5bf8\u548c\u805a\u5408\u7269\u5206\u6563\u6307\u6570\uff08PDI\uff09\uff1b<\/div>\n
\u00a0<\/div>\n
\uff08f\uff09 37 \u2103\u4e0b\uff0cFmoc-H \/ Zn2+<\/sup> \/ Ce6\u548cZ-HF \/ Zn2+<\/sup> \/ Ce6\u5728\u542b\u670910\uff05FBS\u7684PBS\u7f13\u51b2\u6db2\uff08pH=7.4\uff09\u4e2d\u5b75\u80b2\u65f6\u7684\u5c3a\u5bf8\u5927\u5c0f\u548cPDI\uff1b<\/div>\n
\u00a0<\/div>\n
\uff08g\uff09 \u5728\u4e0d\u540c\u7684\u91ca\u653e\u7f13\u51b2\u6db2\u4e2d\uff0cFmoc-H \/ Zn2+<\/sup> \/ Ce6\u4e2d\u7684Ce6\u91ca\u653e\u66f2\u7ebf\u3002<\/div>\n
\u00a0<\/div>\n
\u56fe\u56db\u3001Fmoc-H\/Zn2+<\/sup>\/Ce6\u548cZ-HF\/Zn2+<\/sup>\/Ce6\u5bf9MCF-7\u7684PDT\u4f53\u5916\u8bc4\u4ef7\u00a0\"\"<\/strong><\/div>\n
\u00a0<\/div>\n
\uff08a\uff09 \u4e0e\u91d1\u5c5e\u7eb3\u7c73\u836f\u7269\u8fdb\u884c\u5171\u5b75\u80b2\u540e\u7684\u7ec6\u80deCLSM\u56fe\u50cf\uff0c\u5ef6\u957f\u5b75\u80b2\u65f6\u95f4\u6709\u5229\u4e8e\u7ec6\u80de\u589e\u5f3a\u6444\u53d6\u548c\u91ca\u653e\u91d1\u5c5e\u7eb3\u7c73\u836f\u7269\uff1b<\/div>\n
\u00a0<\/div>\n
\uff08b\uff09 CLSM\u8367\u5149\u56fe\u50cf\u663e\u793aFmoc-H \/ Zn2+<\/sup> \/ Ce6\u5728\u7ec6\u80de\u5185\u7684\u4f4d\u7f6e\uff1b<\/div>\n
\u00a0<\/div>\n
\uff08c\uff09 \u6d41\u5f0f\u7ec6\u80de\u4eea\u6d4b\u5f97\u7684\u7528\u91d1\u5c5e\u7eb3\u7c73\u836f\u7269\u6216\u672a\u5305\u5c01\u7684Ce6\u5b75\u80b2\u540e\u7684\u7ec6\u80de\u8367\u5149\u5f3a\u5ea6\uff1b<\/div>\n
\u00a0<\/div>\n
\uff08d\uff09 \u7ecf\u91d1\u5c5e\u7eb3\u7c73\u836f\u7269\u5b75\u80b2\u548c\u5149\u7167\u5904\u7406\u540e\uff0c\u7ec6\u80de\u4e2dROS\u63a2\u9488\u7684\u8367\u5149\u5f3a\u5ea6\uff1b<\/div>\n
\u00a0<\/div>\n
\uff08e\uff09 CLSM\u56fe\u50cf\u663e\u793a\uff0c\u91d1\u5c5e\u7eb3\u7c73\u836f\u7269\u901a\u8fc7PDT\u4f5c\u7528\u9009\u62e9\u6027\u6740\u4f24\u7ec6\u80de\uff1b<\/div>\n
\u00a0<\/div>\n
\uff08f\uff09 \u901a\u8fc7\u4e0d\u540c\u91d1\u5c5e\u7eb3\u7c73\u836f\u7269\u8fdb\u884cPDT\u540e\u7684\u7ec6\u80de\u6d3b\u6027\u3002<\/div>\n
\u00a0<\/div>\n
\u56fe\u4e94\u3001\u4f53\u5185\u8840\u6db2\u5faa\u73af\u548c\u91d1\u5c5e\u7eb3\u7c73\u836f\u7269\u7684\u751f\u7269\u5206\u5e03\"\"<\/strong><\/div>\n
\u00a0<\/div>\n
\uff08a\uff09 \u9759\u8109\u6ce8\u5c04Fmoc-H \/ Zn2+<\/sup> \/ Ce6\u3001Z-HF \/ Zn2+ <\/sup>\/ Ce6\u6216\u672a\u5305\u5c01\u7684Ce6\u540e\uff0c\u4e0d\u540c\u65f6\u95f4\u70b9\u8840\u6db2\u4e2dCe6\u7684\u6d53\u5ea6\uff1b<\/div>\n
\u00a0<\/div>\n
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\u00a0<\/div>\n
\u6587\u732e\u94fe\u63a5\uff1aSmart Peptide-Based Supramolecular Photodynamic MetalloNanodrugs Designed by Multicomponent Coordination Self-Assembly<\/a><\/strong>\uff08JACS, 2018<\/strong>, DOI: 10.1021\/jacs.8b04912\uff09<\/div>\n
\u00a0<\/div>\n
\u901a\u8baf\u4f5c\u8005\u7b80\u4ecb<\/strong><\/div>\n
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\u8bfe\u9898\u7ec4\u7f51\u7ad9\uff1awww.yan-assembly.org<\/a><\/strong><\/div>\n
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